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MS049 2HCl (1502816-23-0(free base))
CAS No.
MS049 2HCl (1502816-23-0(free base)) ( —— )
Catalog No. M19312 CAS No.
MS049 is a potent and selective inhibitor of PRMT4 (IC50 = 34 nM) and PRMT6 (IC50 = 43 nM).
Purity : 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 47 | Get Quote |
|
| 10MG | 75 | Get Quote |
|
| 25MG | 161 | Get Quote |
|
| 50MG | 303 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameMS049 2HCl (1502816-23-0(free base))
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NoteResearch use only, not for human use.
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Brief DescriptionMS049 is a potent and selective inhibitor of PRMT4 (IC50 = 34 nM) and PRMT6 (IC50 = 43 nM).
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DescriptionMS049 is a potent and selective inhibitor of PRMT4 (IC50 = 34 nM) and PRMT6 (IC50 = 43 nM). It is less active against additional type I PRMTs (IC50s = >130, >220, and 1.6 μM for PRMT1, PRMT3, and PRMT8, respectively) and displays no inhibition against type II or type III PRMTs nor any additional methyltransferases or nonepigenetic targets tested.
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorPRMT4; PRMT6
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Research Area——
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Indication——
Chemical Information
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CAS Number--
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Formula Weight321.28
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Molecular FormulaC15H26Cl2N2O
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Purity98%
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Solubility——
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SMILESCl.Cl.CNCCN1CCC(CC1)OCc2ccccc2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Shen Y, etal. Journal of Medicinal Chemistry, 2016, 59(19):9124-9139.
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