MS049 2HCl (1502816-23-0(free base))

Research use only, not for human use.

MS049 is a potent and selective inhibitor of PRMT4 (IC50 = 34 nM) and PRMT6 (IC50 = 43 nM).

MS049 is a potent and selective inhibitor of PRMT4 (IC50 = 34 nM) and PRMT6 (IC50 = 43 nM). It is less active against additional type I PRMTs (IC50s = >130, >220, and 1.6 μM for PRMT1, PRMT3, and PRMT8, respectively) and displays no inhibition against type II or type III PRMTs nor any additional methyltransferases or nonepigenetic targets tested.

——

Others

Other Targets

PRMT4; PRMT6

——

——

--

321.28

C15H26Cl2N2O

98%

——

Cl.Cl.CNCCN1CCC(CC1)OCc2ccccc2

——

(-20℃)

With Ice Pack

≥ 2 years